Structure–Activity Relationship Studies of the Cyclic Depsipeptide Natural Product YM‐254890, Targeting the Gq Protein H Zhang, XF Xiong, MW Boesgaard, CR Underwood, H Bräuner‐Osborne, ... ChemMedChem 12 (11), 830-834, 2017 | 39 | 2017 |
Structure–activity relationship and conformational studies of the natural product cyclic depsipeptides YM-254890 and FR900359 H Zhang, AL Nielsen, MW Boesgaard, K Harpsøe, NL Daly, XF Xiong, ... European journal of medicinal chemistry 156, 847-860, 2018 | 34 | 2018 |
Structure–Activity Relationship Studies of the Natural Product Gq/11 Protein Inhibitor YM‐254890 XF Xiong, H Zhang, MW Boesgaard, CR Underwood, H Bräuner‐Osborne, ... ChemMedChem 14 (8), 865-870, 2019 | 27 | 2019 |
Selective allosteric antagonists for the G protein-coupled receptor GPRC6A based on the 2-phenylindole privileged structure scaffold H Johansson, MW Boesgaard, L Nørskov-Lauritsen, I Larsen, S Kuhne, ... Journal of Medicinal Chemistry 58 (22), 8938-8951, 2015 | 27 | 2015 |
Delineation of molecular determinants for FR900359 inhibition of Gq/11 unlocks inhibition of Gαs MW Boesgaard, K Harpsøe, M Malmberg, CR Underwood, A Inoue, ... Journal of Biological Chemistry 295 (40), 13850-13861, 2020 | 19 | 2020 |
Structural insight to mutation effects uncover a common allosteric site in class C GPCRs K Harpsøe, MW Boesgaard, C Munk, H Bräuner-Osborne, DE Gloriam Bioinformatics 33 (8), 1116-1120, 2017 | 15 | 2017 |
Identification of Histamine H3 Receptor Ligands Using a New Crystal Structure Fragment-based Method IO Frandsen, MW Boesgaard, K Fidom, AS Hauser, V Isberg, ... Scientific Reports 7 (1), 4829, 2017 | 9 | 2017 |
Chen, Shih-Hsun, 13838 Cheng, Hongqiang, 13798 Chu, Dandan, 13812 Clarkson, Michael W., 13829 S Banerjee, AG Bastian, MW Boesgaard, B Bourgeois, ... | | |