Follow
Krzysztof Z. Łączkowski
Krzysztof Z. Łączkowski
Faculty of Pharmacy, Nicolaus Copernicus University
Verified email at cm.umk.pl
Title
Cited by
Cited by
Year
Discovery of tropinone-thiazole derivatives as potent caspase 3/7 activators, and noncompetitive tyrosinase inhibitors with high antiproliferative activity: Rational design …
K Piechowska, M Świtalska, J Cytarska, K Jaroch, K Łuczykowski, ...
European journal of medicinal chemistry 175, 162-171, 2019
422019
Synthesis, antimicrobial evaluation and theoretical prediction of NMR chemical shifts of thiazole and selenazole derivatives with high antifungal activity against Candida spp.
KZ Łączkowski, K Motylewska, A Baranowska-Łączkowska, A Biernasiuk, ...
Journal of Molecular Structure 1108, 427-437, 2016
342016
Synthesis, antimicrobial activity, and determination of the lipophilicity of ((cyclohex-3-enylmethylene) hydrazinyl) thiazole derivatives
A Biernasiuk, M Kawczyńska, A Berecka-Rycerz, B Rosada, ...
Medicinal Chemistry Research 28, 2023-2036, 2019
332019
Synthesis and in vitro antiproliferative activity of thiazole-based nitrogen mustards: the hydrogen bonding interaction between model systems and nucleobases
K Z Laczkowski, K Misiura, M Switalska, J Wietrzyk, ...
Anti-Cancer Agents in Medicinal Chemistry (Formerly Current Medicinal …, 2014
322014
Benzo [b] thiophene-thiazoles as potent anti-Toxoplasma gondii agents: Design, synthesis, tyrosinase/tyrosine hydroxylase inhibitors, molecular docking study, and antioxidant …
B Rosada, A Bekier, J Cytarska, W Płaziński, O Zavyalova, A Sikora, ...
European Journal of Medicinal Chemistry 184, 111765, 2019
312019
Synthesis, antimicrobial and anticonvulsant screening of small library of tetrahydro-2H-thiopyran-4-yl based thiazoles and selenazoles
KZ Łączkowski, A Biernasiuk, A Baranowska-Łączkowska, S Zielińska, ...
Journal of Enzyme Inhibition and Medicinal Chemistry 31 (sup2), 24-39, 2016
312016
Thiazoles with cyclopropyl fragment as antifungal, anticonvulsant, and anti-Toxoplasma gondii agents: synthesis, toxicity evaluation, and molecular docking study
KZ Łączkowski, N Konklewska, A Biernasiuk, A Malm, K Sałat, A Furgała, ...
Medicinal Chemistry Research 27, 2125-2140, 2018
302018
Synthesis, in vitro biological screening and molecular docking studies of novel camphor-based thiazoles
K Z Laczkowski, K Misiura, A Biernasiuk, A Malm, A Siwek, T Plech, ...
Medicinal Chemistry 10 (6), 600-608, 2014
292014
The ORP basis set designed for optical rotation calculations
A Baranowska‐Łączkowska, KZ Łączkowski
Journal of Computational Chemistry 34 (23), 2006-2013, 2013
292013
Model studies of the optical rotation, and theoretical determination of its sign for β‐pinene and trans‐pinane
A Baranowska, KZ Ła̧czkowski, AJ Sadlej
Journal of computational chemistry 31 (6), 1176-1181, 2010
292010
Synthesis and anticonvulsant activities of novel 2-(cyclopentylmethylene) hydrazinyl-1, 3-thiazoles in mouse models of seizures
KZ Łączkowski, K Sałat, K Misiura, A Podkowa, N Malikowska
Journal of Enzyme Inhibition and Medicinal Chemistry 31 (6), 1576-1582, 2016
282016
The newly synthesized thiazole derivatives as potential antifungal compounds against Candida albicans
A Biernasiuk, A Berecka-Rycerz, A Gumieniczek, M Malm, KZ Łączkowski, ...
Applied Microbiology and Biotechnology 105 (16), 6355-6367, 2021
262021
One-pot telescoped synthesis of thiazole derivatives from β-keto esters and thioureas promoted by tribromoisocyanuric acid
VSC de Andrade, MCS de Mattos
Synthesis 50 (24), 4867-4874, 2018
262018
Thiazole-based nitrogen mustards: design, synthesis, spectroscopic studies, DFT calculation, molecular docking, and antiproliferative activity against selected human cancer …
KZ Łączkowski, M Świtalska, A Baranowska-Łączkowska, T Plech, ...
Journal of Molecular Structure 1119, 139-150, 2016
262016
Synthesis, molecular docking, ctDNA interaction, DFT calculation and evaluation of antiproliferative and anti-Toxoplasma gondii activities of 2,4-diaminotriazine …
KZ Łączkowski, J Anusiak, M Świtalska, K Dzitko, J Cytarska, ...
Medicinal Chemistry Research 27, 1131-1148, 2018
232018
Effect of the dichloro-substitution on antiproliferative activity of phthalimide-thiazole derivatives. Rational design, synthesis, elastase, caspase 3/7, and EGFR tyrosine …
B Donarska, M Świtalska, W Płaziński, J Wietrzyk, KZ Łączkowski
Bioorganic Chemistry 110, 104819, 2021
222021
Tropinone-derived alkaloids as potent anticancer agents: Synthesis, tyrosinase inhibition, mechanism of action, DFT calculation, and molecular docking studies
K Piechowska, M Mizerska-Kowalska, B Zdzisińska, J Cytarska, ...
International Journal of Molecular Sciences 21 (23), 9050, 2020
182020
Asymmetric synthesis of N-substituted N-hydroxyureas
KZ Łączkowski, MM Pakulski, MP Krzemiński, P Jaisankar, M Zaidlewicz
Tetrahedron: Asymmetry 19 (7), 788-795, 2008
182008
Antibacterial Activity, Interaction with Nucleobase and Molecular Docking Studies of 4-Formylbenzoic Acid Based Thiazoles
KZ Łączkowski, A Biernasiuk, A Baranowska-Łączkowska, et al.
Medicinal Chemistry 12, 553-562, 2016
16*2016
Synthesis, antimicrobial activities and molecular docking studies of novel 6-hydroxybenzofuran-3 (2H)-one based 2, 4-disubstituted 1, 3-thiazoles
K Z Laczkowski, K Misiura, A Biernasiuk, A Malm, A Siwek, T Plech
Letters in Drug Design & Discovery 10 (9), 798-807, 2013
162013
The system can't perform the operation now. Try again later.
Articles 1–20