Lipophilicity and Click Reactivity Determine the Performance of Bioorthogonal Tetrazine Tools in Pretargeted In Vivo Chemistry EJL Stéen, JT Jørgensen, C Denk, UM Battisti, K Nørregaard, PE Edem, ... ACS pharmacology & translational science 4 (2), 824-833, 2021 | 62 | 2021 |
DARK classics in chemical neuroscience: NBOMes CBM Poulie, AA Jensen, AL Halberstadt, JL Kristensen ACS chemical neuroscience 11 (23), 3860-3869, 2019 | 51 | 2019 |
Heterocycles as Nonclassical Bioisosteres of α‐Amino Acids CBM Poulie, L Bunch ChemMedChem 8 (2), 205-215, 2013 | 40 | 2013 |
A novel series of histamine H4 receptor antagonists based on the pyrido [3, 2-d] pyrimidine scaffold: comparison of hERG binding and target residence time with PF-3893787 M Andaloussi, HD Lim, T van der Meer, M Sijm, CBM Poulie, IJP de Esch, ... Bioorganic & medicinal chemistry letters 23 (9), 2663-2670, 2013 | 27 | 2013 |
Evaluation of [64Cu]Cu-NOTA-PEG7-H-Tz for Pretargeted Imaging in LS174T Xenografts—Comparison to [111In]In-DOTA-PEG11-BisPy-Tz CBM Poulie, JT Jørgensen, V Shalgunov, G Kougioumtzoglou, ... Molecules 26 (3), 544, 2021 | 25 | 2021 |
One-Step Synthesis of N-Succinimidyl-4-[18F]Fluorobenzoate ([18F]SFB) I Nymann Petersen, J Madsen, C Bernard Matthijs Poulie, A Kjær, ... Molecules 24 (19), 3436, 2019 | 13 | 2019 |
Design, Synthesis, and Pharmacological Characterization of Heterobivalent Ligands for the Putative 5-HT2A/mGlu2 Receptor Complex CBM Poulie, N Liu, AA Jensen, L Bunch Journal of medicinal chemistry 63 (17), 9928-9949, 2020 | 12 | 2020 |
Discovery of β-Arrestin-Biased 25CN-NBOH-Derived 5-HT2A Receptor Agonists CBM Poulie, E Pottie, IA Simon, K Harpsøe, L D’Andrea, IV Komarov, ... Journal of Medicinal Chemistry 65 (18), 12031-12043, 2022 | 10 | 2022 |
The Alkaloids from Lophophora diffusa and Other “False Peyotes” CB Chan, CBM Poulie, SS Wismann, J Soelberg, JL Kristensen Journal of Natural Products 84 (8), 2398-2407, 2021 | 8 | 2021 |
A Diversity Oriented Synthesis Approach to New 2,3-trans-Substituted l-Proline Analogs as Potential Ligands for the Ionotropic Glutamate Receptors S Kayser, P Temperini, CBM Poulie, M Staudt, B Nielsen, DS Pickering, ... ACS Chemical Neuroscience 11 (5), 702-714, 2020 | 8 | 2020 |
Structure–Activity Assessment and In-Depth Analysis of Biased Agonism in a Set of Phenylalkylamine 5-HT2A Receptor Agonists E Pottie, CBM Poulie, IA Simon, K Harpsøe, L D’Andrea, IV Komarov, ... ACS Chemical Neuroscience 14 (15), 2727-2742, 2023 | 7 | 2023 |
Surface adsorption of the alpha-emitter astatine-211 to gold nanoparticles is stable in vivo and potentially useful in radionuclide therapy E Sporer, CBM Poulie, S Lindegren, E Aneheim, H Jensen, T Bäck, ... Journal of Nanotheranostics 2 (4), 196-207, 2021 | 7 | 2021 |
Covalent core-radiolabeling of polymeric micelles with 125I/211At for theranostic radiotherapy E Sporer, CBM Poulie, T Bäck, S Lindegren, H Jensen, PJ Kempen, ... Nanotheranostics 6 (4), 388, 2022 | 6 | 2022 |
Pretargeted theranostics M Staudt, MM Herth, CBM Poulie Theranostics—An Old Concept in New Clothing, 1-19, 2021 | 6 | 2021 |
Bioorthogonal Click of Colloidal Gold Nanoparticles to Antibodies In vivo CBM Poulie, E Sporer, L Hvass, JT Jørgensen, PJ Kempen, ... Chemistry–A European Journal 28 (61), e202201847, 2022 | 4 | 2022 |
Design and Synthesis of 2,3-trans-Proline Analogues as Ligands for Ionotropic Glutamate Receptors and Excitatory Amino Acid Transporters CBM Poulie, A Alcaide, M Krell-Jørgensen, Y Larsen, E Astier, ... ACS chemical neuroscience 10 (6), 2989-3007, 2019 | 4 | 2019 |
Tetrabutylammonium Fluoride as a Mild and Versatile Reagent for Cleaving Boroxazolidones to Their Corresponding Free α‐Amino Acids CBM Poulie, L Bunch European Journal of Organic Chemistry 2017 (11), 1475-1478, 2017 | 4 | 2017 |
Next generation fibroblast activation protein (FAP) targeting PET tracers-The tetrazine ligation allows an easy and convenient way to 18F-labeled (4-quinolinoyl) glycyl-2 … CBM Poulie, V Shalgunov, F Elvas, Y Van Rymenant, ES Moon, ... European Journal of Medicinal Chemistry 262, 115862, 2023 | 2 | 2023 |
(S)-2-Mercaptohistidine: A First Selective Orthosteric GluK3 Antagonist CBM Poulie, Y Larsen, C Leteneur, G Barthet, WE Bjørn-Yoshimoto, ... ACS Chemical Neuroscience 13 (10), 1580-1587, 2022 | 2 | 2022 |
In Vitro and In Vivo Evaluation of Pellotine: A Hypnotic Lophophora Alkaloid CBM Poulie, CB Chan, A Parka, M Lettorp, J Vos, A Raaschou, E Pottie, ... ACS pharmacology & translational science 6 (10), 1492-1507, 2023 | 1 | 2023 |