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Paola Conti
Paola Conti
Professore di Chimica Farmaceutica, Università degli Studi di Milano
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Design of remarkably simple, yet potent urea-based inhibitors of glutamate carboxypeptidase II (NAALADase)
AP Kozikowski, F Nan, P Conti, J Zhang, E Ramadan, T Bzdega, ...
Journal of medicinal chemistry 44 (3), 298-301, 2001
3332001
Synthesis and Biochemical Evaluation of Δ2-Isoxazoline Derivatives as DNA Methyltransferase 1 Inhibitors
S Castellano, D Kuck, M Viviano, J Yoo, F López-Vallejo, P Conti, ...
Journal of medicinal chemistry 54 (21), 7663-7677, 2011
1892011
Synthesis of new Δ2-isoxazoline derivatives and their pharmacological characterization as β-adrenergic receptor antagonists
P Conti, C Dallanoce, M De Amici, C De Micheli, KN Klotz
Bioorganic & medicinal chemistry 6 (4), 401-408, 1998
1271998
Drug discovery targeting amino acid racemases
P Conti, L Tamborini, A Pinto, A Blondel, P Minoprio, A Mozzarelli, ...
Chemical reviews 111 (11), 6919-6946, 2011
1242011
Inhibition of rhodesain as a novel therapeutic modality for human African trypanosomiasis
R Ettari, L Tamborini, IC Angelo, N Micale, A Pinto, C De Micheli, P Conti
Journal of Medicinal Chemistry 56 (14), 5637-5658, 2013
982013
A regioselective route to 5-substituted pyrazole-and pyrazoline-3-phosphonic acids and esters
P Conti, A Pinto, L Tamborini, V Rizzo, C De Micheli
Tetrahedron 63 (25), 5554-5560, 2007
882007
The glial glutamate transporter 1 (GLT1) is expressed by pancreatic β-cells and prevents glutamate-induced β-cell death
ES Di Cairano, AM Davalli, L Perego, S Sala, VF Sacchi, S La Rosa, ...
Journal of Biological Chemistry 286 (16), 14007-14018, 2011
782011
UCP2 inhibition induces ROS/Akt/mTOR axis: Role of GAPDH nuclear translocation in genipin/everolimus anticancer synergism
I Dando, R Pacchiana, E Dalla Pozza, I Cataldo, S Bruno, P Conti, ...
Free Radical Biology and Medicine 113, 176-189, 2017
602017
An efficient method for the lipase-catalysed resolution and in-line purification of racemic flurbiprofen in a continuous-flow reactor
L Tamborini, D Romano, A Pinto, A Bertolani, F Molinari, P Conti
Journal of Molecular Catalysis B: Enzymatic 84, 78-82, 2012
592012
Synthesis and functional characterization of novel derivatives related to oxotremorine and oxotremorine-M
C Dallanoce, P Conti, M De Amici, C De Micheli, E Barocelli, M Chiavarini, ...
Bioorganic & medicinal chemistry 7 (8), 1539-1547, 1999
581999
Synthesis, binding affinity at glutamic acid receptors, neuroprotective effects, and molecular modeling investigation of novel dihydroisoxazole amino acids
P Conti, M De Amici, G Grazioso, G Roda, A Pinto, KB Hansen, B Nielsen, ...
Journal of medicinal chemistry 48 (20), 6315-6325, 2005
572005
Discovery of covalent inhibitors of glyceraldehyde-3-phosphate dehydrogenase, a target for the treatment of malaria
S Bruno, A Pinto, G Paredi, L Tamborini, C De Micheli, V La Pietra, ...
Journal of Medicinal Chemistry 57 (17), 7465-7471, 2014
552014
An efficient continuous flow process for the synthesis of a non-conventional mixture of fructooligosaccharides
P Zambelli, L Tamborini, S Cazzamalli, A Pinto, S Arioli, S Balzaretti, ...
Food Chemistry 190, 607-613, 2016
522016
Chemoenzymatic synthesis in flow reactors: A rapid and convenient preparation of Captopril
V De Vitis, F Dall'Oglio, A Pinto, C De Micheli, F Molinari, P Conti, ...
ChemistryOpen 6 (5), 668-673, 2017
502017
Design and synthesis of novel isoxazole-based HDAC inhibitors
P Conti, L Tamborini, A Pinto, L Sola, R Ettari, C Mercurio, C De Micheli
European journal of medicinal chemistry 45 (9), 4331-4338, 2010
502010
Mutant p53 prevents GAPDH nuclear translocation in pancreatic cancer cells favoring glycolysis and 2-deoxyglucose sensitivity
G Butera, R Pacchiana, N Mullappilly, M Margiotta, S Bruno, P Conti, ...
Biochimica et Biophysica Acta (BBA)-Molecular Cell Research 1865 (12), 1914-1923, 2018
492018
Flow-based stereoselective reduction of ketones using an immobilized ketoreductase/glucose dehydrogenase mixed bed system
F Dall'Oglio, ML Contente, P Conti, F Molinari, D Monfredi, A Pinto, ...
Catalysis Communications 93, 29-32, 2017
492017
Synthesis and enantiopharmacology of new AMPA-kainate receptor agonists
P Conti, M De Amici, G De Sarro, M Rizzo, TB Stensbøl, ...
Journal of medicinal chemistry 42 (20), 4099-4107, 1999
481999
Development of rhodesain inhibitors with a 3‐bromoisoxazoline warhead
R Ettari, L Tamborini, IC Angelo, S Grasso, T Schirmeister, L Lo Presti, ...
ChemMedChem 8 (12), 2070-2076, 2013
452013
Biotransformation with whole microbial systems in a continuous flow reactor: resolution of (RS)-flurbiprofen using Aspergillus oryzae by direct esterification with ethanol in …
L Tamborini, D Romano, A Pinto, M Contente, MC Iannuzzi, P Conti, ...
Tetrahedron letters 54 (45), 6090-6093, 2013
432013
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